Avaliação da umbeliferona e seus derivados substituídos como potenciais inibidores da enzima GST-π e determinação de seus perfies farmacocinéticos via estudos in silico
Resumo
The inhibitory activity of coumarins against glutathione-S-transferase was assessed by molecular docking. Docking results suggest a greater inhibitory potential of compounds 3 and 6. In general, pharmacokinetic requirements were met for coumarins. However, toxicity must be improved.
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Publicado
2019-07-24
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Ciências da saúde